Journal article Open access Published 2025

Identification of a novel Azaspirooxindolinone-based PROTAC for selective BTK degradation and enhanced anticancer activity

N.K. Rampeesa, R. Gundla, G. Mudasani, S. Tangallapalli, S.R. Anugu, Soňa Gurská, Juan Bautista De Sanctis, Petr Džubák, Marián Hajdúch, Viswanath Das

Bioorganic Chemistry 157, 108316 (2025)

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RAMPEESA, N., R. GUNDLA, G. MUDASANI, S. TANGALLAPALLI, S. ANUGU, S. GURSKÁ, J. DE SANCTIS, P. DŽUBÁK, M. HAJDÚCH, V. DAS: Identification of a novel Azaspirooxindolinone-based PROTAC for selective BTK degradation and enhanced anticancer activity. Bioorganic Chemistry. 2025, 157, 108316, ISSN: 0045-2068, PMID: 40037026,  PDF.

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